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Discovery of a Highly Selective Cell-Active Inhibitor of the Histone Lysine Demethylases KDM2/7
Gerken, P.A., Wolstenhulme, J.R., Tumber, A., Hatch, S.B., Zhang, Y., Müller, S., Chandler, S.A., Mair, B., Li, F., Nijman, S.M.B., Konietzny, R., Szommer, T., Yapp, C., Fedorov, O., Benesch, J.L.P., Vedadi, M., Kessler, B.M., Kawamura, A., Brennan, P.E., Smith, M.D.
Angew. Chem. (International ed. in English) (2017), 56 (49), 15555-15559
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